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Two Birds with One Stone: A Novel Dithiomaleimide-Based GalNAc-siRNA Conjugate Enabling Good siRNA Delivery and Traceability

For the first time, a novel dithiomaleimides (DTM) based tetra-antennary GalNAc conjugate was developed, which enable both efficient siRNA delivery and good traceability, without incorporating extra fluorophores. This conjugate can be readily constructed by three click-type reactions, that is, amida...

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Principais autores: Sudong Kong, Xiaoqing Gao, Qianhui Wang, Jianguo Lin, Ling Qiu, Minhao Xie
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI AG 2023-10-01
coleção:Molecules
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Acesso em linha:https://www.mdpi.com/1420-3049/28/20/7184
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