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Is asciminib an effective tyrosine kinase inhibitor for chronic myeloid leukemia patients with tyrosine kinase inhibitor resistance?

Asciminib represents a significant advancement in the treatment of chronic myeloid leukemia, establishing a novel therapeutic paradigm by specifically targeting the ABL1 myristoyl pocket, a mechanism distinct from that of conventional adenosine triphosphate-competitive inhibitors. Such a selective i...

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Detaylı Bibliyografya
Asıl Yazarlar: Musab MA Omar, Majed A Alanazi, Denise E. Jackson
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Elsevier 2026-04-01
Seri Bilgileri:Hematology, Transfusion and Cell Therapy
Konular:
Online Erişim:http://www.sciencedirect.com/science/article/pii/S2531137926000040
Etiketler: Etiketle
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