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Biopharmaceutical and pharmacokinetic attributes to drive nanoformulations of small molecule tyrosine kinase inhibitors

Buoyed by the discovery of small-molecule tyrosine kinase inhibitors (smTKIs), significant impact has been made in cancer chemotherapeutics. However, some of these agents still encounter off-target toxicities and suboptimal efficacies due to their inferior biopharmaceutical and/or pharmacokinetic pr...

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Autori principali: Soumyadip Mukherjee, Vedant Joshi, Kolimi Prashanth Reddy, Nidhi Singh, Priyanka Das, Pallab Datta
Natura: Artigo
Lingua:Inglês
Pubblicazione: KeAi Communications Co., Ltd. 2024-12-01
Serie:Asian Journal of Pharmaceutical Sciences
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Accesso online:http://www.sciencedirect.com/science/article/pii/S1818087624000977
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