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Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (<i>Pseudo</i>)-Dipeptidyl Appendages: In Vitro and Computational Studies

The involvement of human carbonic anhydrase (hCA) IX/XII in the pathogenesis and progression of many types of cancer is well acknowledged, and more recently human monoamine oxidases (hMAOs) A and B have been found important contributors to tumor development and aggressiveness. With a view of an enzy...

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Autori principali: Mariangela Agamennone, Marialuigia Fantacuzzi, Simone Carradori, Anél Petzer, Jacobus P. Petzer, Andrea Angeli, Claudiu T. Supuran, Grazia Luisi
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI AG 2022-11-01
Serie:Molecules
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Accesso online:https://www.mdpi.com/1420-3049/27/22/7884
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