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Mipsagargin: The Beginning—Not the End—of Thapsigargin Prodrug-Based Cancer Therapeutics

Søren Brøgger Christensen isolated and characterized the cell-penetrant sesquiterpene lactone Thapsigargin (TG) from the fruit <i>Thapsia garganica.</i> In the late 1980s/early 1990s, TG was supplied to multiple independent and collaborative groups. Using this TG, studies documented with a large var...

Ausführliche Beschreibung

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Bibliografische Detailangaben
Hauptverfasser: John T. Isaacs, William Nathaniel Brennen, Søren Brøgger Christensen, Samuel R. Denmeade
Format: Artigo
Sprache:Inglês
Veröffentlicht: MDPI AG 2021-12-01
Schriftenreihe:Molecules
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Online-Zugang:https://www.mdpi.com/1420-3049/26/24/7469
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