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Bicyclic Basic Merbarone Analogues as Antiproliferative Agents

Pyrimido-pyrimidine derivatives have been developed as rigid merbarone analogues. In a previous study, these compounds showed potent antiproliferative activity and efficiently inhibited topoisomerase IIα. To further extend the structure–activity relationships on pyrimido-pyrimidines, a novel series...

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Bibliografiske detaljer
Principais autores: Andrea Spallarossa, Matteo Lusardi, Chiara Caneva, Aldo Profumo, Camillo Rosano, Marco Ponassi
Format: Artigo
Sprog:Inglês
Udgivet: MDPI AG 2021-01-01
Serier:Molecules
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Online adgang:https://www.mdpi.com/1420-3049/26/3/557
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