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Revisiting capsaicin and nonivamide: Their analogs exert strong inhibitory activity against cholinesterases

The scientific community has long been interested in capsaicin, and the extensive hunt for AChE and BChE enzyme inhibitors is still ongoing. In this investigation analogs of capsaicin, such as the pharmaceutical nonivamide, which is preferred in clinical settings for the topical treatment of pain, w...

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Autori principali: Niels V. Heise, Jeremy Quast, René Csuk
Natura: Artigo
Lingua:Inglês
Pubblicazione: Elsevier 2024-12-01
Serie:European Journal of Medicinal Chemistry Reports
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Accesso online:http://www.sciencedirect.com/science/article/pii/S2772417424000724
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