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Comparative evaluation for small molecule somatostatin 4 receptor agonists: in silico, in vitro, and in vivo approaches

IntroductionThe treatment of neuropathic pain with traditional and adjuvant analgesics is limited in efficacy and associated with severe adverse effects. Our group has previously shown that somatostatin, released from capsaicin-sensitive peptidergic sensory nerve terminals, mediates analgesic and an...

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Autors principals: Dóra Biskup, Minjin Ganbold, Andrea Kinga Nehr-Majoros, Valéria Tékus, Zsófia Hajna, Barbara Fülöp, Éva Szőke, Csaba Hetényi, A. Michael Crider, Iman Daryaei, Zsuzsanna Helyes, Rita Börzsei, Erika Pintér
Format: Artigo
Idioma:Inglês
Publicat: Frontiers Media S.A. 2026-06-01
Col·lecció:Frontiers in Pharmacology
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Accés en línia:https://www.frontiersin.org/articles/10.3389/fphar.2026.1838782/full
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