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Structural insights into the orthosteric inhibition of P2X receptors by non-ATP analog antagonists

P2X receptors are extracellular ATP-gated ion channels that form homo- or heterotrimers and consist of seven subtypes. They are expressed in various tissues, including neuronal and nonneuronal cells, and play critical roles in physiological processes such as neurotransmission, inflammation, pain, an...

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Principais autores: Danqi Sheng, Chen-Xi Yue, Fei Jin, Yao Wang, Muneyoshi Ichikawa, Ye Yu, Chang-Run Guo, Motoyuki Hattori
Formato: Artigo
Idioma:Inglês
Publicado: eLife Sciences Publications Ltd 2024-04-01
Series:eLife
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Acceso en liña:https://elifesciences.org/articles/92829
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