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Comparison of gepant effects at therapeutic plasma concentrations: connecting pharmacodynamics and pharmacokinetics

Abstract Background Orally administered second-generation gepants are effective for the treatment of migraine. The intranasal administration of the third-generation gepant zavegepant might have additional benefits including a rapid onset of action, but it is not clear yet to which extent this has cl...

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Autores principales: Deirdre M. Boucherie, Ruben Dammers, Arnaud Vincent, A. H. Jan Danser, Antoinette MaassenVanDenBrink
Formato: Artigo
Lenguaje:Inglês
Publicado: BMC 2024-08-01
Colección:The Journal of Headache and Pain
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Acceso en línea:https://doi.org/10.1186/s10194-024-01846-8
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