Biased allosteric agonism and modulation of metabotropic glutamate receptor 5: implications for optimizing preclinical neuroscience drug discovery

著者: Sengmany, Kathy, Singh, Junaid, Stewart, Gregory D., Conn, P. Jeffrey, Christopoulos, Arthur, Gregory, Karen J.
出版年 Neuropharmacology (2016)

Kinetic and system bias as drivers of metabotropic glutamate receptor 5 allosteric modulator pharmacology

著者: Sengmany, Kathy, Hellyer, Shane D., Albold, Sabine, Wang, Taide, Jeffrey Conn, P., May, Lauren T., Christopoulos, Arthur, Leach, Katie, Gregory, Karen J.
出版年 Neuropharmacology (2019)