Pharmacological characterization of potent and selective Na(V)1.7 inhibitors engineered from Chilobrachys jingzhao tarantula venom peptide JzTx-V

von Moyer, Bryan D., Murray, Justin K., Ligutti, Joseph, Andrews, Kristin, Favreau, Philippe, Jordan, John B., Lee, Josie H., Liu, Dong, Long, Jason, Sham, Kelvin, Shi, Licheng, Stöcklin, Reto, Wu, Bin, Yin, Ruoyuan, Yu, Violeta, Zou, Anruo, Biswas, Kaustav, Miranda, Les P.
Veröffentlicht in PLoS One (2018)

Sulfonamides as Selective Na(V)1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement

von Marx, Isaac E., Dineen, Thomas A., Able, Jessica, Bode, Christiane, Bregman, Howard, Chu-Moyer, Margaret, DiMauro, Erin F., Du, Bingfan, Foti, Robert S., Fremeau, Robert T., Gao, Hua, Gunaydin, Hakan, Hall, Brian E., Huang, Liyue, Kornecook, Thomas, Kreiman, Charles R., La, Daniel S., Ligutti, Joseph, Lin, Min-Hwa Jasmine, Liu, Dong, McDermott, Jeff S., Moyer, Bryan D., Peterson, Emily A., Roberts, Jonathan T., Rose, Paul, Wang, Jean, Youngblood, Beth D., Yu, Violeta, Weiss, Matthew M.
Veröffentlicht in ACS Med Chem Lett (2016)

Correction to “Sulfonamides as Selective Na(V)1.7 Inhibitors: Optimizing Potency and Pharmacokinetics to Enable in Vivo Target Engagement”

von Marx, Isaac E., Dineen, Thomas A., Able, Jessica, Bode, Christiane, Bregman, Howard, Chu-Moyer, Margaret, DiMauro, Erin F., Du, Bingfan, Foti, Robert S., Fremeau, Robert T., Gao, Hua, Gunaydin, Hakan, Hall, Brian E., Huang, Liyue, Kornecook, Thomas, Kreiman, Charles R., La, Daniel S., Ligutti, Joseph, Lin, Min-Hwa Jasmine, Liu, Dong, McDermott, Jeff S., Moyer, Bryan D., Nguyen, Hanh N., Peterson, Emily A., Roberts, Jonathan T., Rose, Paul, Wang, Jean, Youngblood, Beth D., Yu, Violeta, Weiss, Matthew M.
Veröffentlicht in ACS Med Chem Lett (2017)