Oxopyrido[2,3-d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors

著者: Wurz, Ryan P., Pettus, Liping H., Ashton, Kate, Brown, James, Chen, Jian Jeffrey, Herberich, Brad, Hong, Fang-Tsao, Hu-Harrington, Essa, Nguyen, Tom, St. Jean, David J., Tadesse, Seifu, Bauer, David, Kubryk, Michele, Zhan, Jinghui, Cooke, Keegan, Mitchell, Petia, Andrews, Kristin L., Hsieh, Faye, Hickman, Dean, Kalyanaraman, Nataraj, Wu, Tian, Reid, Darren L., Lobenhofer, Edward K., Andrews, Dina A., Everds, Nancy, Guzman, Roberto, Parsons, Andrew T., Hedley, Simon J., Tedrow, Jason, Thiel, Oliver R., Potter, Matthew, Radinsky, Robert, Beltran, Pedro J., Tasker, Andrew S.
出版年 ACS Med Chem Lett (2015)