Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors

по Serafini, Marta, Torre, Enza, Aprile, Silvio, Massarotti, Alberto, Fallarini, Silvia, Pirali, Tracey
Опубликовано в: Molecules (2019)

Data on metabolic stability, aqueous solubility and CYP inhibition of novel triazole-based nicotinamide phosphoribosyltransferase (NAMPT) inhibitors

по Aprile, Silvio, Galli, Ubaldina, Tron, Gian Cesare, Del Grosso, Erika, Travelli, Cristina, Grosa, Giorgio
Опубликовано в: Data Brief (2019)

Biological effects of combined resveratrol and vitamin D3 on ovarian tissue

по Uberti, Francesca, Morsanuto, Vera, Aprile, Silvio, Ghirlanda, Sabrina, Stoppa, Ian, Cochis, Andrea, Grosa, Giorgio, Rimondini, Lia, Molinari, Claudio
Опубликовано в: J Ovarian Res (2017)

1,2,4-Oxadiazole-Bearing Pyrazoles as Metabolically Stable Modulators of Store-Operated Calcium Entry

по Aprile, Silvio, Riva, Beatrice, Bhela, Irene Preet, Cordero-Sanchez, Celia, Avino, Giulia, Genazzani, Armando A., Serafini, Marta, Pirali, Tracey
Опубликовано в: ACS Med Chem Lett (2021)

Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors

по Serafini, Marta, Cordero-Sanchez, Celia, Di Paola, Rosanna, Bhela, Irene P., Aprile, Silvio, Purghè, Beatrice, Fusco, Roberta, Cuzzocrea, Salvatore, Genazzani, Armando A., Riva, Beatrice, Pirali, Tracey
Опубликовано в: J Med Chem (2020)

Identification of a Potent Phosphoinositide 3‐Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs

по Pirali, Tracey, Ciraolo, Elisa, Aprile, Silvio, Massarotti, Alberto, Berndt, Alex, Griglio, Alessia, Serafini, Marta, Mercalli, Valentina, Landoni, Clarissa, Campa, Carlo Cosimo, Margaria, Jean Piero, Silva, Rangel L., Grosa, Giorgio, Sorba, Giovanni, Williams, Roger, Hirsch, Emilio, Tron, Gian Cesare
Опубликовано в: ChemMedChem (2017)

Inhalation of the prodrug PI3K inhibitor CL27c improves lung function in asthma and fibrosis

по Campa, Carlo C., Silva, Rangel L., Margaria, Jean P., Pirali, Tracey, Mattos, Matheus S., Kraemer, Lucas R., Reis, Diego C., Grosa, Giorgio, Copperi, Francesca, Dalmarco, Eduardo M., Lima-Júnior, Roberto C. P., Aprile, Silvio, Sala, Valentina, Dal Bello, Federica, Prado, Douglas Silva, Alves-Filho, Jose Carlos, Medana, Claudio, Cassali, Geovanni D., Tron, Gian Cesare, Teixeira, Mauro M., Ciraolo, Elisa, Russo, Remo C., Hirsch, Emilio
Опубликовано в: Nat Commun (2018)