Synthesis, Docking and Biological Evaluation of a Novel Class of Imidazothiazoles as IDO1 Inhibitors

par Serafini, Marta, Torre, Enza, Aprile, Silvio, Massarotti, Alberto, Fallarini, Silvia, Pirali, Tracey
Publié dans Molecules (2019)

Data on metabolic stability, aqueous solubility and CYP inhibition of novel triazole-based nicotinamide phosphoribosyltransferase (NAMPT) inhibitors

par Aprile, Silvio, Galli, Ubaldina, Tron, Gian Cesare, Del Grosso, Erika, Travelli, Cristina, Grosa, Giorgio
Publié dans Data Brief (2019)

Biological effects of combined resveratrol and vitamin D3 on ovarian tissue

par Uberti, Francesca, Morsanuto, Vera, Aprile, Silvio, Ghirlanda, Sabrina, Stoppa, Ian, Cochis, Andrea, Grosa, Giorgio, Rimondini, Lia, Molinari, Claudio
Publié dans J Ovarian Res (2017)

1,2,4-Oxadiazole-Bearing Pyrazoles as Metabolically Stable Modulators of Store-Operated Calcium Entry

par Aprile, Silvio, Riva, Beatrice, Bhela, Irene Preet, Cordero-Sanchez, Celia, Avino, Giulia, Genazzani, Armando A., Serafini, Marta, Pirali, Tracey
Publié dans ACS Med Chem Lett (2021)

Store-Operated Calcium Entry as a Therapeutic Target in Acute Pancreatitis: Discovery and Development of Drug-Like SOCE Inhibitors

par Serafini, Marta, Cordero-Sanchez, Celia, Di Paola, Rosanna, Bhela, Irene P., Aprile, Silvio, Purghè, Beatrice, Fusco, Roberta, Cuzzocrea, Salvatore, Genazzani, Armando A., Riva, Beatrice, Pirali, Tracey
Publié dans J Med Chem (2020)

Identification of a Potent Phosphoinositide 3‐Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs

par Pirali, Tracey, Ciraolo, Elisa, Aprile, Silvio, Massarotti, Alberto, Berndt, Alex, Griglio, Alessia, Serafini, Marta, Mercalli, Valentina, Landoni, Clarissa, Campa, Carlo Cosimo, Margaria, Jean Piero, Silva, Rangel L., Grosa, Giorgio, Sorba, Giovanni, Williams, Roger, Hirsch, Emilio, Tron, Gian Cesare
Publié dans ChemMedChem (2017)

Inhalation of the prodrug PI3K inhibitor CL27c improves lung function in asthma and fibrosis

par Campa, Carlo C., Silva, Rangel L., Margaria, Jean P., Pirali, Tracey, Mattos, Matheus S., Kraemer, Lucas R., Reis, Diego C., Grosa, Giorgio, Copperi, Francesca, Dalmarco, Eduardo M., Lima-Júnior, Roberto C. P., Aprile, Silvio, Sala, Valentina, Dal Bello, Federica, Prado, Douglas Silva, Alves-Filho, Jose Carlos, Medana, Claudio, Cassali, Geovanni D., Tron, Gian Cesare, Teixeira, Mauro M., Ciraolo, Elisa, Russo, Remo C., Hirsch, Emilio
Publié dans Nat Commun (2018)