Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors

Por Morteza Abdoli, Murat Bozdag, Andrea Angeli, Claudiu T. Supuran
Publicado em 2018-06-01

Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII

Por Andrea Angeli, Fabio Vaiano, Francesco Mari, Elisabetta Bertol, Claudiu T. Supuran
Publicado em 2017-01-01

Synthesis of a new series of 3-functionalised-1-phenyl-1,2,3-triazole sulfamoylbenzamides as carbonic anhydrase I, II, IV and IX inhibitors

Por Baijayantimala Swain, Andrea Angeli, Srinivas Angapelly, Pavitra S. Thacker, Priti Singh, Claudiu T. Supuran, Mohammed Arifuddin
Publicado em 2019-01-01

Fluoroenesulphonamides: N-sulphonylurea isosteres showing nanomolar selective cancer-related transmembrane human carbonic anhydrase inhibition

Por Benoit Métayer, Andrea Angeli, Agnès Mingot, Kévin Jouvin, Gwilherm Evano, Claudiu T. Supuran, Sébastien Thibaudeau
Publicado em 2018-01-01

Synthesis and Biological Evaluation of Imidazo[2,1-<i>b</i>]Thiazole based Sulfonyl Piperazines as Novel Carbonic Anhydrase II Inhibitors

Por Kesari Lakshmi Manasa, Sravya Pujitha, Aaftaab Sethi, Mohammed Arifuddin, Mallika Alvala, Andrea Angeli, Claudiu T. Supuran
Publicado em 2020-03-01

Design, Synthesis, and Biological Evaluation of 1,2,3-Triazole-Linked Triazino[5,6-B]Indole-Benzene Sulfonamide Conjugates as Potent Carbonic Anhydrase I, II, IX, and XIII Inhibito...

Por Krishna Kartheek Chinchilli, Andrea Angeli, Pavitra S. Thacker, Laxman Naik Korra, Rashmita Biswas, Mohammed Arifuddin, Claudiu T. Supuran
Publicado em 2020-05-01

The first activation study of a δ-carbonic anhydrase: TweCAδ from the diatom Thalassiosira weissflogii is effectively activated by amines and amino acids

Por Andrea Angeli, Fatmah A. S. Alasmary, Sonia Del Prete, Sameh M. Osman, Zeid AlOthman, William A. Donald, Clemente Capasso, Claudiu T. Supuran
Publicado em 2018-01-01

Activation of β- and γ-carbonic anhydrases from pathogenic bacteria with tripeptides

Por Azzurra Stefanucci, Andrea Angeli, Marilisa Pia Dimmito, Grazia Luisi, Sonia Del Prete, Clemente Capasso, William A. Donald, Adriano Mollica, Claudiu T. Supuran
Publicado em 2018-01-01

Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases

Por Giannamaria Annunziato, Laura Giovati, Andrea Angeli, Marialaura Pavone, Sonia Del Prete, Marco Pieroni, Clemente Capasso, Agostino Bruno, Stefania Conti, Walter Magliani, Claudiu T. Supuran, Gabriele Costantino
Publicado em 2018-01-01

Evaluation of Thio- and Seleno-Acetamides Bearing Benzenesulfonamide as Inhibitor of Carbonic Anhydrases from Different Pathogenic Bacteria

Por Andrea Angeli, Mariana Pinteala, Stelian S. Maier, Bogdan C. Simionescu, Andrea Milaneschi, Ghulam Abbas, Sonia del Prete, Clemente Capasso, Antonella Capperucci, Damiano Tanini, Fabrizio Carta, Claudiu T. Supuran
Publicado em 2020-01-01

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold

Por Giulia Rotondi, Paolo Guglielmi, Simone Carradori, Daniela Secci, Celeste De Monte, Barbara De Filippis, Cristina Maccallini, Rosa Amoroso, Roberto Cirilli, Atilla Akdemir, Andrea Angeli, Claudiu T. Supuran
Publicado em 2019-01-01

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment

Por Andrea Angeli, Fabrizio Carta, Alessio Nocentini, Jean-Yves Winum, Raivis Zalubovskis, Atilla Akdemir, Valentina Onnis, Wagdy M. Eldehna, Clemente Capasso, Giuseppina De Simone, Simona Maria Monti, Simone Carradori, William A. Donald, Shoukat Dedhar, Claudiu T. Supuran
Publicado em 2020-10-01