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Unveiling the “invisible” druggable conformations of GDP-bound inactive Ras

The prevalent view on whether Ras is druggable has gradually changed in the recent decade with the discovery of effective inhibitors binding to cryptic sites unseen in the native structures. Despite the promising advances, therapeutics development toward higher potency and specificity is challenged...

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Podrobná bibliografie
Vydáno v:Proc Natl Acad Sci U S A
Hlavní autoři: Liu, Dan, Mao, Yunyun, Gu, Xue, Zhou, Yang, Long, Dong
Médium: Artigo
Jazyk:Inglês
Vydáno: National Academy of Sciences 2021
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7980447/
https://ncbi.nlm.nih.gov/pubmed/33836610
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.2024725118
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