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A solid lipid nanoparticle formulation of 4-(N)-docosahexaenoyl 2′, 2′-difluorodeoxycytidine with increased solubility, stability, and antitumor activity

Previously, we synthesized 4-(N)-docosahexaenoyl 2′, 2′-difluorodeoxycytidine (DHA-dFdC), a novel lipophilic compound with a potent, broad-spectrum antitumor activity. Herein, we report a solid lipid nanoparticle (SLN) formulation of DHA-dFdC with improved apparent aqueous solubility, chemical stabi...

詳細記述

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書誌詳細
出版年:Int J Pharm
主要な著者: Valdes, Solange A., Alzhrani, Riyad F., Rodriguez, Andres, Lansakara-P, Dharmika S.P., Thakkar, Sachin G., Cui, Zhengrong
フォーマット: Artigo
言語:Inglês
出版事項: 2019
主題:
オンライン・アクセス:https://ncbi.nlm.nih.gov/pmc/articles/PMC6824728/
https://ncbi.nlm.nih.gov/pubmed/31415878
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ijpharm.2019.118609
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