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Homology Model and Docking-Based Virtual Screening for Ligands of Human Dyskerin as New Inhibitors of Telomerase for Cancer Treatment

Immortality is one of the main features of cancer cells. Tumor cells have an unlimited replicative potential, principally due to the holoenzyme telomerase. Telomerase is composed mainly by dyskerin (DKC1), a catalytic retrotranscriptase (hTERT) and an RNA template (hTR). The aim of this work is to d...

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Dettagli Bibliografici
Pubblicato in:Int J Mol Sci
Autori principali: Armando, Romina Gabriela, Mengual Gómez, Diego Luis, Juritz, Ezequiel Ivan, Lorenzano Menna, Pablo, Gomez, Daniel Eduardo
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6214037/
https://ncbi.nlm.nih.gov/pubmed/30340325
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms19103216
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