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The E(2.65)A mutation disrupts dynamic binding poses of SB269652 at the dopamine D2 and D3 receptors

The dopamine D2 and D3 receptors (D2R and D3R) are important targets for antipsychotics and for the treatment of drug abuse. SB269652, a bitopic ligand that simultaneously binds both the orthosteric binding site (OBS) and a secondary binding pocket (SBP) in both D2R and D3R, was found to be a negati...

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Publicat a:PLoS Comput Biol
Autors principals: Verma, Ravi Kumar, Abramyan, Ara M., Michino, Mayako, Free, R. Benjamin, Sibley, David R., Javitch, Jonathan A., Lane, J. Robert, Shi, Lei
Format: Artigo
Idioma:Inglês
Publicat: Public Library of Science 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5786319/
https://ncbi.nlm.nih.gov/pubmed/29337986
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pcbi.1005948
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