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Identification of 5-Nitrofuran-2-Amide Derivatives that Induce Apoptosis in Triple Negative Breast Cancer Cells by Activating C/EBP-Homologous Protein Expression

The transcription factor C/EBP-homologous protein (CHOP) is a key component of the terminal unfolded protein response (UPR) that mediates unresolvable endoplasmic reticulum stress-induced apoptosis. CHOP induction is known to cause cancer cell death. Chemicals that induce CHOP expression would thus...

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Библиографические подробности
Опубликовано в: :Bioorg Med Chem
Главные авторы: Duan, Hongliang, Li, Yu, Lim, Hui-Ying, Wang, Weidong
Формат: Artigo
Язык:Inglês
Опубликовано: 2015
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5567983/
https://ncbi.nlm.nih.gov/pubmed/26116180
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2015.06.011
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