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ADP inhibits function of the ABC transporter cystic fibrosis transmembrane conductance regulator via its adenylate kinase activity

ADP interacts with the nucleotide-binding domains (NBDs) of the cystic fibrosis transmembrane conductance regulator (CFTR) to inhibit its Cl(-) channel activity. Because CFTR NBD2 has reversible adenylate kinase activity (ATP + AMP ⇆ ADP + ADP) that gates the channel, we asked whether ADP might inhi...

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Detaylı Bibliyografya
Asıl Yazarlar: Randak, Christoph O., Welsh, Michael J.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: National Academy of Sciences 2005
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC548590/
https://ncbi.nlm.nih.gov/pubmed/15684079
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0409787102
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