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Crizotinib (PF02341066) as a ALK /MET inhibitor— Special Emphasis as a Therapeutic Drug Against Lung Cancer

There are a number of molecular abnormalities that can occur in normal cells to induce a malignant phenotype. Recently, the receptor tyrosine kinase anaplastic lymphoma kinase (ALK) has been shown to have gain-of-function when partnered with different proteins. As an example, on chromosome 2p, with...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Drugs Future
Prif Awduron: Nwizu, Tobenna, Kanteti, Rajani, Kawada, Ichiro, Rolle, Cleo, Vokes, Everett E., Salgia, Ravi
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2011
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC4582997/
https://ncbi.nlm.nih.gov/pubmed/26412935
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1358/dof.2011.036.02.1584112
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