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Time Resolved Fluorescence Resonance Energy Transfer Assay for Discovery of Small Molecule Inhibitors of Methyl-CpG Binding Domain Protein 2

Methylated DNA binding proteins such as Methyl-CpG Binding Domain Protein 2 (MBD2) can transduce DNA methylation alterations into a repressive signal by recruiting transcriptional co-repressor complexes. Interfering with MBD2 could lead to re-activation of tumor suppressor genes and therefore repres...

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Autori principali: Wyhs, Nicolas, Walker, David, Giovinazzo, Hugh, Yegnasubramanian, Srinivasan, Nelson, William G
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4183726/
https://ncbi.nlm.nih.gov/pubmed/24608100
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1177/1087057114526433
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