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Click Chemistry in Peptide-Based Drug Design

Click chemistry is an efficient and chemoselective synthetic method for coupling molecular fragments under mild reaction conditions. Since the advent in 2001 of methods to improve stereochemical conservation, the click chemistry approach has been broadly used to construct diverse chemotypes in both...

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Autors principals: Li, Huiyuan, Aneja, Rachna, Chaiken, Irwin
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2013
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4155329/
https://ncbi.nlm.nih.gov/pubmed/23959192
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules18089797
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