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Efficient Traceless Solid-Phase Synthesis of 3,4-Dihydropyrazino[1,2-b]indazoles and their 6-Oxides
A highly efficient novel traceless solid-phase synthesis of 3,4-dihydropyrazino[1,2-b]indazoles and their 6-oxides was developed by using commercially available building blocks, diamines, 2-nitrobenzenesulfonyl chlorides, and bromoketones/bromoacetates. Mild reaction conditions, diversely substitute...
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Autors principals: | , |
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Format: | Artigo |
Idioma: | Inglês |
Publicat: |
2009
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Matèries: | |
Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC2703815/ https://ncbi.nlm.nih.gov/pubmed/19245249 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cc800181y |
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