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Functions of Acidic Transmembrane Residues in Human Melanocortin-3 Receptor Binding and Activation

The melanocortin-3 receptor (MC3R) is an important regulator of energy homeostasis, inflammation, and cardiovascular function. Inactivating mutations in MC3R gene are associated with childhood obesity. How MC3R binds to its ligands has rarely been studied. In the present study, we systematically mut...

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Autori principali: Wang, Shu-Xiu, Fan, Zhen-Chuan, Tao, Ya-Xiong
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2008
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC2536753/
https://ncbi.nlm.nih.gov/pubmed/18614155
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2008.05.026
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