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Redefining the structure-activity relationships of 2,6-methano-3-benzazocines. 6. Opioid receptor binding properties of cyclic variants of 8-carboxamidocyclazocine

A series of 7,8- and 8,9-fused pyrimidinone, aminopyridine and pyridone derivatives of 8-carboxamidocyclazocine (8-CAC) have been prepared and evaluated in opioid receptor binding assays. Targets were designed to corroborate a pharmacophore hypothesis regarding the bioactive conformation of the carb...

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Détails bibliographiques
Auteurs principaux: Wentland, Mark P., Sun, Xufeng, Cohen, Dana J., Bidlack, Jean M.
Format: Artigo
Langue:Inglês
Publié: 2008
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC2441872/
https://ncbi.nlm.nih.gov/pubmed/18417347
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2008.03.066
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