Synthesis and Antiplasmodial Evaluation of 4-Carboxamido- and 4-Alkoxy-2-Trichloromethyl Quinazolines

por Amrane, Dyhia, Gellis, Armand, Hutter, Sébastien, Prieri, Marion, Verhaeghe, Pierre, Azas, Nadine, Vanelle, Patrice, Primas, Nicolas
Publicado en Molecules (2020)

A New Synthetic Route to Original Sulfonamide Derivatives in 2-Trichloromethylquinazoline Series: A Structure-Activity Relationship Study of Antiplasmodial Activity

por Primas, Nicolas, Verhaeghe, Pierre, Cohen, Anita, Kieffer, Charline, Dumètre, Aurélien, Hutter, Sébastien, Rault, Sylvain, Rathelot, Pascal, Azas, Nadine, Vanelle, Patrice
Publicado en Molecules (2012)

In Vitro Evaluation of the Antiviral Activity of Methylene Blue Alone or in Combination against SARS-CoV-2

por Gendrot, Mathieu, Jardot, Priscilla, Delandre, Océane, Boxberger, Manon, Andreani, Julien, Duflot, Isabelle, Le Bideau, Marion, Mosnier, Joel, Fonta, Isabelle, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Publicado en J Clin Med (2021)

Antimalarial artemisinin-based combination therapies (ACT) and COVID-19 in Africa: In vitro inhibition of SARS-CoV-2 replication by mefloquine-artesunate

por Gendrot, Mathieu, Duflot, Isabelle, Boxberger, Manon, Delandre, Océane, Jardot, Priscilla, Le Bideau, Marion, Andreani, Julien, Fonta, Isabelle, Mosnier, Joel, Rolland, Clara, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Publicado en Int J Infect Dis (2020)

Antimalarial drugs inhibit the replication of SARS-CoV-2: An in vitro evaluation

por Gendrot, Mathieu, Andreani, Julien, Boxberger, Manon, Jardot, Priscilla, Fonta, Isabelle, Le Bideau, Marion, Duflot, Isabelle, Mosnier, Joel, Rolland, Clara, Bogreau, Hervé, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Publicado en Travel Med Infect Dis (2020)

Methylene blue inhibits replication of SARS-CoV-2 in vitro

por Gendrot, Mathieu, Andreani, Julien, Duflot, Isabelle, Boxberger, Manon, Le Bideau, Marion, Mosnier, Joel, Jardot, Priscilla, Fonta, Isabelle, Rolland, Clara, Bogreau, Hervé, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Publicado en Int J Antimicrob Agents (2020)

In Vitro Antiviral Activity of Doxycycline against SARS-CoV-2

por Gendrot, Mathieu, Andreani, Julien, Jardot, Priscilla, Hutter, Sébastien, Delandre, Océane, Boxberger, Manon, Mosnier, Joel, Le Bideau, Marion, Duflot, Isabelle, Fonta, Isabelle, Rolland, Clara, Bogreau, Hervé, La Scola, Bernard, Pradines, Bruno
Publicado en Molecules (2020)

Novel 8-nitroquinolin-2(1H)-ones as NTR-bioactivated antikinetoplastid molecules: Synthesis, electrochemical and SAR study

por Pedron, Julien, Boudot, Clotilde, Hutter, Sébastien, Bourgeade-Delmas, Sandra, Stigliani, Jean-Luc, Sournia-Saquet, Alix, Moreau, Alain, Boutet-Robinet, Elisa, Paloque, Lucie, Mothes, Emmanuelle, Laget, Michèle, Vendier, Laure, Pratviel, Geneviève, Wyllie, Susan, Fairlamb, Alan, Azas, Nadine, Courtioux, Bertrand, Valentin, Alexis, Verhaeghe, Pierre
Publicado en Eur J Med Chem (2018)

8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases

por Fersing, Cyril, Boudot, Clotilde, Pedron, Julien, Hutter, Sébastien, Primas, Nicolas, Castera-Ducros, Caroline, Bourgeade-Delmas, Sandra, Sournia-Saquet, Alix, Moreau, Alain, Cohen, Anita, Stigliani, Jean-Luc, Pratviel, Geneviève, Crozet, Maxime D., Wyllie, Susan, Fairlamb, Alan, Valentin, Alexis, Rathelot, Pascal, Azas, Nadine, Courtioux, Bertrand, Verhaeghe, Pierre, Vanelle, Patrice
Publicado en Eur J Med Chem (2018)

Nongenotoxic 3-Nitroimidazo[1,2-a]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial Activity

por Fersing, Cyril, Basmaciyan, Louise, Boudot, Clotilde, Pedron, Julien, Hutter, Sébastien, Cohen, Anita, Castera-Ducros, Caroline, Primas, Nicolas, Laget, Michèle, Casanova, Magali, Bourgeade-Delmas, Sandra, Piednoel, Mélanie, Sournia-Saquet, Alix, Belle Mbou, Valère, Courtioux, Bertrand, Boutet-Robinet, Élisa, Since, Marc, Milne, Rachel, Wyllie, Susan, Fairlamb, Alan H., Valentin, Alexis, Rathelot, Pascal, Verhaeghe, Pierre, Vanelle, Patrice, Azas, Nadine
Publicado en ACS Med Chem Lett (2018)