Synthesis and Antiplasmodial Evaluation of 4-Carboxamido- and 4-Alkoxy-2-Trichloromethyl Quinazolines

von Amrane, Dyhia, Gellis, Armand, Hutter, Sébastien, Prieri, Marion, Verhaeghe, Pierre, Azas, Nadine, Vanelle, Patrice, Primas, Nicolas
Veröffentlicht in Molecules (2020)

A New Synthetic Route to Original Sulfonamide Derivatives in 2-Trichloromethylquinazoline Series: A Structure-Activity Relationship Study of Antiplasmodial Activity

von Primas, Nicolas, Verhaeghe, Pierre, Cohen, Anita, Kieffer, Charline, Dumètre, Aurélien, Hutter, Sébastien, Rault, Sylvain, Rathelot, Pascal, Azas, Nadine, Vanelle, Patrice
Veröffentlicht in Molecules (2012)

In Vitro Evaluation of the Antiviral Activity of Methylene Blue Alone or in Combination against SARS-CoV-2

von Gendrot, Mathieu, Jardot, Priscilla, Delandre, Océane, Boxberger, Manon, Andreani, Julien, Duflot, Isabelle, Le Bideau, Marion, Mosnier, Joel, Fonta, Isabelle, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Veröffentlicht in J Clin Med (2021)

Antimalarial artemisinin-based combination therapies (ACT) and COVID-19 in Africa: In vitro inhibition of SARS-CoV-2 replication by mefloquine-artesunate

von Gendrot, Mathieu, Duflot, Isabelle, Boxberger, Manon, Delandre, Océane, Jardot, Priscilla, Le Bideau, Marion, Andreani, Julien, Fonta, Isabelle, Mosnier, Joel, Rolland, Clara, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Veröffentlicht in Int J Infect Dis (2020)

Antimalarial drugs inhibit the replication of SARS-CoV-2: An in vitro evaluation

von Gendrot, Mathieu, Andreani, Julien, Boxberger, Manon, Jardot, Priscilla, Fonta, Isabelle, Le Bideau, Marion, Duflot, Isabelle, Mosnier, Joel, Rolland, Clara, Bogreau, Hervé, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Veröffentlicht in Travel Med Infect Dis (2020)

Methylene blue inhibits replication of SARS-CoV-2 in vitro

von Gendrot, Mathieu, Andreani, Julien, Duflot, Isabelle, Boxberger, Manon, Le Bideau, Marion, Mosnier, Joel, Jardot, Priscilla, Fonta, Isabelle, Rolland, Clara, Bogreau, Hervé, Hutter, Sébastien, La Scola, Bernard, Pradines, Bruno
Veröffentlicht in Int J Antimicrob Agents (2020)

In Vitro Antiviral Activity of Doxycycline against SARS-CoV-2

von Gendrot, Mathieu, Andreani, Julien, Jardot, Priscilla, Hutter, Sébastien, Delandre, Océane, Boxberger, Manon, Mosnier, Joel, Le Bideau, Marion, Duflot, Isabelle, Fonta, Isabelle, Rolland, Clara, Bogreau, Hervé, La Scola, Bernard, Pradines, Bruno
Veröffentlicht in Molecules (2020)

Novel 8-nitroquinolin-2(1H)-ones as NTR-bioactivated antikinetoplastid molecules: Synthesis, electrochemical and SAR study

von Pedron, Julien, Boudot, Clotilde, Hutter, Sébastien, Bourgeade-Delmas, Sandra, Stigliani, Jean-Luc, Sournia-Saquet, Alix, Moreau, Alain, Boutet-Robinet, Elisa, Paloque, Lucie, Mothes, Emmanuelle, Laget, Michèle, Vendier, Laure, Pratviel, Geneviève, Wyllie, Susan, Fairlamb, Alan, Azas, Nadine, Courtioux, Bertrand, Valentin, Alexis, Verhaeghe, Pierre
Veröffentlicht in Eur J Med Chem (2018)

8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases

von Fersing, Cyril, Boudot, Clotilde, Pedron, Julien, Hutter, Sébastien, Primas, Nicolas, Castera-Ducros, Caroline, Bourgeade-Delmas, Sandra, Sournia-Saquet, Alix, Moreau, Alain, Cohen, Anita, Stigliani, Jean-Luc, Pratviel, Geneviève, Crozet, Maxime D., Wyllie, Susan, Fairlamb, Alan, Valentin, Alexis, Rathelot, Pascal, Azas, Nadine, Courtioux, Bertrand, Verhaeghe, Pierre, Vanelle, Patrice
Veröffentlicht in Eur J Med Chem (2018)

Nongenotoxic 3-Nitroimidazo[1,2-a]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial Activity

von Fersing, Cyril, Basmaciyan, Louise, Boudot, Clotilde, Pedron, Julien, Hutter, Sébastien, Cohen, Anita, Castera-Ducros, Caroline, Primas, Nicolas, Laget, Michèle, Casanova, Magali, Bourgeade-Delmas, Sandra, Piednoel, Mélanie, Sournia-Saquet, Alix, Belle Mbou, Valère, Courtioux, Bertrand, Boutet-Robinet, Élisa, Since, Marc, Milne, Rachel, Wyllie, Susan, Fairlamb, Alan H., Valentin, Alexis, Rathelot, Pascal, Verhaeghe, Pierre, Vanelle, Patrice, Azas, Nadine
Veröffentlicht in ACS Med Chem Lett (2018)